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Purpose
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A potent and selective protease-activated receptor 2 (PAR2) agonist
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Characteristics
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AC 55541 is a potent and selective protease-activated receptor 2 (PAR2) agonist (pEC?? = 6.7) that displays no activity at other PAR subtypes or at over 30 other receptors involved in nociception and inflammation.
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Purity
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≥ 98?% by HPLC
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Chemical Name
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2E)-2-[1-(3-Bromophenyl)ethylidene] α-(benzoylamino)-3,4-dihydro-4-oxo-1-phthalazineacetic acid hydrazide
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Formula
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C??H??BrN?O?
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Permeability
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Cell-permeable
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Solubility
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DMSO (~ 25 mg/ml)
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